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UNC 9994 hydrochloride
UNC 9994 hydrochloride
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  • 商品货号:A16087
  • 名称:UNC 9994 hydrochloride
  • 简介:UNC 9994 hydrochloride, unique, beta-arrestin-biased functionally selective dopamine D2 receptor (D2R) agonist (Ki value 30 nM; EC50 value 50 nM in ??-arrestin-2 recruitment assay) that exhibits antipsychotic activity in vivo. UNC9994 markedly inhibited PCP-induced hyperlocomotion in wild-type mice, which effect was completely abolished in ??-arrestin-2 knockout mice.
  • CASNO:1354030-51-5
  • 分子式:C21H23Cl3N2OS
  • 分子量:457.84
  • SMILES:C1CN(CCC1C2=C(C(=CC=C2)Cl)Cl)CCCOC3=CC4=C(C=C3)SC=N4.Cl
  • 保持条件:at -20°C 3 years Powder
  • 同名:UNC9994 hydrochloride
  • 纯度:>98%
  • 应用:dopamine D2 receptor agonist
  • 作用机制:Agonist