- 名称:Evacetrapib (LY2484595)
- 简介:Evacetrapib (LY2484595) is a potent and selective inhibitor of CETP with IC50 of 5.5 nM, elevates HDL cholesterol without increases in aldosterone or blood pressure. Phase 3.
- CASNO:1186486-62-3
- 分子式:C31H36F6N6O2
- 分子量:638.65
- SMILES:CC1=CC(=C2C(=C1)[C@H](CCCN2CC3CCC(CC3)C(=O)O)N(CC4=CC(=CC(=C4)C(F)(F)F)C(F)(F)F)C5=NN(N=N5)C)C
- 保持条件:at -20°C 3 years Powder
- 同名:LY2484595, LY-2484595, LY 2484595
- 纯度:>98%
- 应用:CETP inhibitor
- 作用机制:Inhibitor