• 名称：GSK126
• 简介：GSK126 is a potent, highly selective, S-adenosyl-methionine-competitive, small-molecule inhibitor of EZH2 methyltransferase activity, decreases global H3K27me3 levels and reactivates silenced PRC2 target genes.
• CASNO：1346574-57-9
• 分子式：C31H38N6O2
• 分子量：526.67
• SMILES：CC[C@H](C)N1C=C(C2=C(C=C(C=C21)C3=CN=C(C=C3)N4CCNCC4)C(=O)NCC5=C(C=C(NC5=O)C)C)C
• 保持条件：at -20°C 3 years Powder
• 同名：GSK 126, GSK-126
• 纯度：>98%
• 应用：EZH2 inhibitor
• 作用机制：Inhibitor