- 名称:SR 144528
- 简介:SR 144528 is a selective peripheral cannabinoid receptor inverse agonist that displays a Ki value of 0.6 nM for rat spleen and human recombinant CB2 receptors and a Ki value of 400 nM for rat brain and human recombinant CB1 receptors.
- CASNO:192703-06-3
- 分子式:C29H34ClN3O
- 分子量:476.05
- SMILES:CC1=CC=C(C=C1)CN2C(=CC(=N2)C(=O)N[C@H]3[C@]4(CC[C@H](C4)C3(C)C)C)C5=CC(=C(C=C5)Cl)C
- 保持条件:at -20°C 3 years Powder
- 同名:SR144528, SR-144528
- 纯度:>98%
- 应用:CB2 inverse agonist
- 作用机制:Agonist