- 名称:EPZ-6438 (Tazemetostat)
- 简介:EPZ-6438 is a potent, selective, and orally bioavailable small-molecule inhibitor of EZH2 enzymatic activity. It induces apoptosis and differentiation specifically in SMARCB1-deleted MRT cells.
- CASNO:1403254-99-8
- 分子式:C34H44N4O4
- 分子量:572.74
- SMILES:CCN(C1CCOCC1)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C4=CC=C(C=C4)CN5CCOCC5
- 保持条件:at -20°C 3 years Powder
- 同名:EPZ6438, EPZ 6438
- 纯度:>98%
- 应用:EZH2 inhibitor
- 作用机制:Inhibitor