- 名称:GSK221149A (Retosiban)
- 简介:Retosiban (GSK-221,149-A) is an oral drug which acts as a selective, sub-nanomolar (Ki = 0.65 nM) oxytocin receptor antagonist with >1400-fold selectivity over the related vasopressin receptors
- CASNO:820957-38-8
- 分子式:C27H34N4O5
- 分子量:494.58
- SMILES:CC[C@H](C)[C@@H]1C(=O)N[C@@H](C(=O)N1[C@H](C2=COC(=N2)C)C(=O)N3CCOCC3)C4CC5=CC=CC=C5C4
- 保持条件:at -20°C 3 years Powder
- 同名:GSK-221149A, GSK 221149A
- 纯度:>98%
- 应用:Oxytocin Receptor Antagonist
- 作用机制:Antagonist