- 名称:GSK2656157
- 简介:GSK2656157 is an ATP-competitive inhibitor of PERK enzyme activity with an IC(50) of 0.9 nmol/L. It is highly selective for PERK with IC(50) values >100 nmol/L against a panel of 300 kinases.
- CASNO:1337532-29-2
- 分子式:C23H21FN6O
- 分子量:416.45
- SMILES:CC1=NC(=CC=C1)CC(=O)N2CCC3=C2C=CC(=C3F)C4=CN(C5=C4C(=NC=N5)N)C
- 保持条件:at -20°C 3 years Powder
- 同名:GSK 2656157
- 纯度:>98%
- 应用:PERK Inhibitor
- 作用机制:Inhibitor