- 名称:JNJ-10397049
- 简介:JNJ-10397049 is a potent, selective, and bioavailable antagonist of the orexin-2 receptor (OX2R) (KB = 4.5 nM for OX2R versus 1.1 μM for OX1R).
- CASNO:708275-58-5
- 分子式:C19H20Br2N2O3
- 分子量:484.2
- SMILES:CC1(OC[C@@H]([C@@H](O1)C2=CC=CC=C2)NC(=O)NC3=C(C=C(C=C3)Br)Br)C
- 保持条件:at -20°C 3 years Powder
- 同名:JNJ 10397049, JNJ10397049
- 纯度:>98%
- 应用:OX2 receptor antagonist
- 作用机制:Antagonist