- 名称:Tedalinab
- 简介:Tedalinab (GRC-10693) is a drug developed for the treatment of osteoarthritis and neuropathic pain, which acts as a potent and selective cannabinoid CB2 receptor agonist. It has a very high selectivity of 4700x for CB2 over the related CB1 receptor, has good oral bioavailability and has shown promising safety results and effective analgesic and antiinflammatory actions in early clinical trials.
- CASNO:916591-01-0
- 分子式:C19H21F2N3O
- 分子量:345.4
- SMILES:CC(C)(C)NC(=O)C1=NN(C2=C1[C@H]3CC[C@@H]2C3)C4=C(C=C(C=C4)F)F
- 保持条件:at -20°C 3 years Powder
- 同名:GRC-10693
- 纯度:>98%
- 应用:CB2 receptor agonist
- 作用机制:Agonist