- 名称:PF-06463922
- 简介:PF-06463922 is a potent, dual ALK/ROS1 inhibitor with Ki of <0.02 nM, <0.07 nM, and 0.7 nM for ROS1, ALK (WT), and ALK (L1196M), respectively.
- CASNO:1454846-35-5
- 分子式:C21H19FN6O2
- 分子量:406.41
- SMILES:C[C@@H]1C2=C(C=CC(=C2)F)C(=O)N(CC3=NN(C(=C3C4=CC(=C(N=C4)N)O1)C#N)C)C
- 保持条件:at -20°C 3 years Powder
- 同名:PF 06463922, PF06463922
- 纯度:>98%
- 应用:ALK inhibitor
- 作用机制:Inhibitor