- 名称:PFI-2
- 简介:PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
- CASNO:1627676-59-8
- 分子式:C23H25F4N3O3S
- 分子量:499.52
- SMILES:C1CCN(C1)C(=O)[C@@H](CC2=CC(=CC=C2)C(F)(F)F)NS(=O)(=O)C3=CC(=C4CNCCC4=C3)F
- 保持条件:at -20°C 3 years Powder
- 同名:PFI2
- 纯度:>98%
- 应用:SETD7 inhibitor
- 作用机制:Inhibitor