• 名称：TRV130 (Oliceridine)
• 简介：TRV130 is an opioid drug that is under evaluation in human clinical trials for the treatment of acute severe pain. TRV130 elicits robust G protein signaling, with potency and efficacy similar to morphine, but with far less ??-arrestin 2 recruitment and receptor internalization, it displays less adverse effects than morphine.
• CASNO：1401028-24-7
• 分子式：C22H31ClN2O2S
• 分子量：423.01
• SMILES：COC1=C(SC=C1)CNCC[C@]2(CCOC3(C2)CCCC3)C4=CC=CC=N4
• 保持条件：at -20°C 3 years Powder
• 同名：TRV 130, TRV-130
• 纯度：>98%
• 应用：μ-opioid receptor agonist
• 作用机制：Agonist