- 名称:GSK256066 2,2,2-trifluoroacetic acid
- 简介:GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.
- CASNO:1415560-64-3
- 分子式:C29H27F3N4O7S
- 分子量:632.61
- SMILES:CC1=C2C(=CC(=C1)S(=O)(=O)C3=CC=CC(=C3)C(=O)N(C)C)C(=C(C=N2)C(=O)N)NC4=CC(=CC=C4)OC.C(=O)(C(F)(F)F)O
- 保持条件:at -20°C 3 years Powder
- 同名:GSK-256066, GSK 256066
- 纯度:>98%
- 应用:PDE Inhibitor
- 作用机制:Inhibitor