- 名称:TRV130 HCl (Oliceridine)
- 简介:TRV 130 HCl is a novel μ-opioid receptor (MOR) G protein-biased ligand; elicits robust G protein signaling(pEC50=8.1), with potency and efficacy similar to morphine, but with far less beta-arrestin recruitment and receptor internalization.
- CASNO:1401031-39-7
- 分子式:C22H31ClN2O2S
- 分子量:423.01
- SMILES:COC1=C(SC=C1)CNCCC2(CCOC3(C2)CCCC3)C4=CC=CC=N4.Cl
- 保持条件:at -20°C 3 years Powder
- 同名:TRV-130, TRV 130
- 纯度:>98%
- 应用:?- opioid receptor agonist
- 作用机制:Agonist