- 名称:WDR5-0103
- 简介:WDR5-0103 is a small molecule that binds a peptide-binding pocket on WDR5 (Kd = 450 nM), inhibiting the catalytic activity of the MLL core complex in vitro (IC50 = 39 M).
- CASNO:890190-22-4
- 分子式:C21H25N3O4
- 分子量:383.45
- SMILES:O=C(OC)C1=CC(NC(C2=CC=CC(OC)=C2)=O)=C(N3CCN(C)CC3)C=C1
- 保持条件:at -20°C 3 years Powder
- 同名:WDR 5-0103, WDR-5-0103
- 纯度:>98%
- 应用:WDR5 antagonist
- 作用机制:Antagonist