• 名称：GSK 5959
• 简介：GSK 5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor with IC50 ~ 80 nM. Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
• CASNO：901245-65-6
• 分子式：C22H26N4O3
• 分子量：394.48
• SMILES：O=C(NC1=C(N2CCCCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
• 保持条件：at -20°C 3 years Powder
• 同名：GSK-5959, GSK5959
• 纯度：>98%
• 应用：BRPF1 bromodomain inhibitor
• 作用机制：Inhibitor