• 名称：TSU-68 (Orantinib, SU6668)
• 简介：Orantinib (TSU-68, SU6668) has greatest potency against PDGFR autophosphorylation with Ki of 8 nM in a cell-free assay, but also strongly inhibits Flk-1 and FGFR1 trans-phosphorylation, little activity against IGF-1R, Met, Src, Lck, Zap70, Abl and CDK2; does not inhibit EGFR. Phase 3.
• CASNO：252916-29-3
• 分子式：C18H18N2O3
• 分子量：310.4
• SMILES：CC1=C(NC(=C1CCC(=O)O)C)/C=C2/C3=CC=CC=C3NC2=O
• 保持条件：at -20°C 3 years Powder
• 同名：TSU68
• 纯度：>98%
• 应用：PDFGRβ inhibitor
• 作用机制：Inhibitor