- 名称:PF299804 (Dacomitinib, PF299)
- 简介:PF299804 is a potent, orally available, irreversible inhibitor of tyrosine kinase human epidermal growth factor receptors (HER) 1 (EGFR), HER2, and HER4.
- CASNO:1110813-31-4
- 分子式:C24H25ClFN5O2
- 分子量:469.9
- SMILES:COC1=C(C=C2C(=C1)N=CN=C2NC3=CC(=C(C=C3)F)Cl)NC(=O)/C=C/CN4CCCCC4
- 保持条件:at -20°C 3 years Powder
- 同名:PF-299804, Dacomitinib, PF-299
- 纯度:>98%
- 应用:EGFR inhibitor
- 作用机制:Inhibitor